Towards the understanding of halogenation in peptide hydrogels: a quantum chemical approach.
Bettens, T.; Lacanau, V.; Van Lommel, R.; De Maeseneer, T.; Vandeplassche, W.; Brancart, J.; Barlow, T.; Woller, T. M.; Van den Brande, N.; Moldenaers, P.; De Proft, F.; Madder, A.; Hoogenboom, R.; Martin, C.; Ballet, S.; Alonso Giner, M. Materials Advances, 2021 2(14), 4792-4803.
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Towards the understanding of halogenation in peptide hydrogels: a quantum chemical approach.
Bettens, T.; Lacanau, V.; Van Lommel, R.; De Maeseneer, T.; Vandeplassche, W.; Brancart, J.; Barlow, T.; Woller, T. M.; Van den Brande, N.; Moldenaers, P.; De Proft, F.; Madder, A.; Hoogenboom, R.; Martin, C.; Ballet, S.; Alonso Giner, M. Materials Advances, 2021 2(14), 4792-4803.
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Brønsted Acid-Catalyzed Enantioselective Iodocycloetherification Enabled by Triphenylphosphine Selenide Cocatalysis
Guria, S.; Daniliuc, C.G.; Hennecke, U.; Adv. Synth. Catal. 2021, 363, 3852-3858.
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3-Substituted 2-isocyanopyridines as versatile convertible isocyanides for peptidomimetic design
Hollanders, C.; Elsocht, M.; Van der Poorten, O.; Jida, M.; Renders, E.; Maes, B.U.W.; Ballet, S. Chem Comm, 2021, DOI: 10.1039/D1CC01701B...
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Antinociceptive Efficacy of the μ‐Opioid/Nociceptin Peptide‐Based Hybrid KGNOP1 in Inflammatory Pain without Rewarding Effects in Mice: An Experimental Assessment and Molecular Docking
Dumitrascuta, M.; Bermudez, M.; Trovato, O.; Neve, J.D.; Ballet, S.; Wolber, G.; Spetea, M., Molecules 2021, 26, 3267.
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A dynamic picture of the halolactonization reaction through a combination of ab initio metadynamics and experimental investigations
R. Van Lommel, J. Bock, C.G. Daniliuc, U. Hennecke, F. De Proft, Chem. Sci. 2021, DOI: 10.1039/D1SC01014J.
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Using conformational constraints at position 6 of Angiotensin II to generate compounds with enhanced AT2R selectivity and proteolytic stability
Tourwé, D.; Tsiailanis, A. D.; Parisis, N.; Hirmiz, B.; Del Borgo, M.; Aguilar, M.-I.; Van der Poorten, O.; Ballet, S.; Widdop, R. E.;Tzakos, A. G., Bioorg. Med. Chem. Lett, 2021, 43, 128086.
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Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors
De Neve, J.; Barlow, T. M.; Tourwé, D.; Bihel, F.; Simonin, F.; Ballet, S., RSC Med. Chem., 2021 DIO: 10.1039/D1MD00041A...
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New review on biased ligand for opiod receptors made the cover
We are pleased to announce that our review has been featured on the cover of RCS Medicinal Chemistry. For a full read, please visit the publisher's page
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Antinociceptive Efficacy of the µ-Opioid/Nociceptin Peptide-Based Hybrid KGNOP1 in Inflammatory Pain without Rewarding Effects in Mice: An Experimental Assessment and Molecular Docking
Dumitrascuta, M.; Bermudez, M.; Trovato, O.; De Neve, J.; Ballet, S.; Wolber, G.; Spetea, M.
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Modification of the Pseudomonas aeruginosa toxin 2-heptyl-1-hydroxyquinolin-4(1H)-one and other secondary metabolites by methyltransferases from mycobacteria
P. Sartor, J. Bock, U. Hennecke, S. Thierbach, S. Fetzner, FEBS J. 2021, 288, 2360-2376.
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Enantioselective Dihalogenation of Alkenes
U. Hennecke, J. Bock, S. Guria, V. Wedek, Chem. Eur. J. 2021, 27, 4517-4530.
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